pkpd.Release0.1.0 package

Model Fitting and Simulation for Drug Release Kinetics and PK/PD

first_order_release

First-Order Drug Release Kinetic Model

higuchi_release

Higuchi Drug Release Kinetic Model

hixson_crowell_model

Hixson-Crowell Drug Release Kinetic Model

korsmeyer_peppas_model

Korsmeyer-Peppas Drug Release Kinetic Model

one_compartment_iv_bolus

One-Compartment IV Bolus Pharmacokinetic Model (Linear)

weibull_model

Weibull Drug Release Kinetic Model

zero_order_release

Zero-Order Drug Release Kinetic Model

ld50_model

Lethal Dose 50 (LD50) Pharmacodynamic Model

logistic_4pl

4PL Logistic Dose-Response Model (Emax/Imax)

logistic_5pl

5PL Logistic Dose-Response Model (Emax/Imax, Asymmetric)

michaelis_menten_nl

Michaelis-Menten Kinetics (Nonlinear Form) with Inhibition Comparison

michaelis_menten

Michaelis-Menten Kinetics (Linear Form) with Inhibition Comparison

non_compartmental_nl

Non-Compartmental Analysis (NCA) of Plasma Concentration-Time Data (No...

non_compartmental

Non-Compartmental Analysis (NCA) of Plasma Concentration-Time Data (Li...

one_compartment_iv_bolus_nl

One-Compartment IV Bolus Pharmacokinetic Model (Nonlinear)

one_compartment_oral_nl

One-Compartment Oral Pharmacokinetic Model (Nonlinear, First-Order Abs...

one_compartment_oral

One-Compartment Oral Pharmacokinetic Model (Linear, First-Order Absorp...

sigmoid_emax

Sigmoid Emax (Stimulatory Hill Model) for Dose-Response Analysis

sigmoid_imax

Sigmoid Imax (Inhibitory Hill Model) for Dose-Response Analysis

td50_model

Toxic Dose 50 (TD50) Pharmacodynamic Model

two_compartment_iv_bolus_nl

Two-Compartment IV Bolus Pharmacokinetic Model (Nonlinear)

two_compartment_iv_bolus

Two-Compartment IV Bolus Pharmacokinetic Model (Linear)

Provides a comprehensive framework for model fitting and simulation of drug release kinetics, pharmacokinetics (PK), and pharmacodynamics (PD). The package implements widely used mechanistic and empirical models for in vitro drug release, including zero-order, first-order, Higuchi, Korsmeyer-Peppas, Hixson-Crowell, and Weibull models. Pharmacokinetic functionality includes linear and nonlinear functions for one- and two-compartment models for intravenous bolus and oral administration, Michaelis-Menten kinetics, and non-compartmental analysis (NCA). Pharmacodynamic and dose-response modeling is supported through Emax-based models, including stimulatory (sigmoid Emax) and inhibitory (sigmoid Imax) Hill models, four- and five-parameter logistic models, as well as median toxic dose (TD50) and lethal dose (LD50) models. The package is intended to support parameter estimation, simulation, and model comparison in pharmaceutical research, drug development, and pharmacometrics education. For more details, see Gabrielsson & Weiner (2000) <ISBN:9186274929>, Holford & Sheiner (1981) <doi:10.2165/00003088-198106060-00002>, and Manlapaz (2025) <doi:10.32614/CRAN.package.adsoRptionCMF>.

  • Maintainer: Paul Angelo C. Manlapaz
  • License: GPL-3
  • Last published: 2026-01-27